Taw qhia thiab daim ntawv thov CAS:285983-48-4|Doramapimod
BIRB 796 (Doramapimod) yog ib qho kev xaiv p38 MAPK inhibitor nrog Kd ntawm 0.1 nM. Nws yog 330 lub sij hawm xaiv ntau dua li JNK2. Nws tsis muaj zog tiv thaiv c-RAF, Fyn thiab Lck, thiab tseem tsis muaj zog tiv thaiv ERK-1 thiab SYK. , IKK2, ZAP-70, EGFR, HER2, PKA, PKC, PKC / / .
Specification of CAS: 285983-48-4|Doramapimod
| Yam khoom | Specification |
Melting point: 142-143 degree
Kub taw tes: 631.6 ± 55.0 degree (Predicted)
Qhov ceev: 1.2 0± 0.1g / cm3 (Tshaj tawm)
Cia tej yam kev mob: Sealedindry, Storeinfreezer, nyob rau hauv -20 degree
Solubility: Soluble hauv DMSO (txog 50mg / ml) lossis ethanol (txog 30mg / ml).
Daim ntawv: khov
Acidity coefficient (pKa): 13.47 ± 0.70 (Predicted)
Xim: dawb los yog tawm-dawb
Pob thiab kev thauj mus los ntawm CAS: 285983-48-4|Doramapimod
Kev thauj mus los: los ntawm courier / los ntawm huab cua / los ntawm hiav txwv.
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